Home

helps physicians and healthcare professionals

Erectile Dysfunction

helps physicians and healthcare professionals

Doctor123.org

helps physicians and healthcare professionals

Hydroxyamphetamine and Tropicamide


General


Pronunciation

(hye droks ee am FET a meen & troe PIK a mide)


Brand Names: U.S.

  • Paremyd

Indications


Use: Labeled Indications

Mydriasis: Short-term pupil dilation for diagnostic procedures


Contraindications


Hypersensitivity to hydroxyamphetamine, tropicamide, or any component of the formulation; angle-closure glaucoma or those with narrow angles where dilation of the pupil may precipitate angle-closure glaucoma


Dosing and Administration


Dosing: Adult

Mydriasis: Ophthalmic: Instill 1 to 2 drops into conjunctival sac(s)


Dosing: Geriatric

Refer to adult dosing.


Dosing: Renal Impairment

There are no dosage adjustments provided in manufacturer 's labeling.


Dosing: Hepatic Impairment

There are no dosage adjustments provided in manufacturer 's labeling.


Administration

For topical ophthalmic use only. To avoid excessive systemic absorption, apply gentle finger pressure to lacrimal sac for 2 to 3 minutes following application. Do not touch dropper tip to eyelids or other surfaces when placing drops in eyes. Wash hands following administration.


Storage

Store between 20 ‚ °C and 25 ‚ °C (68 ‚ °F and 77 ‚ °F). Protect from light. Protect from light.


Dosage Forms/Strengths


Dosage Forms

Excipient information presented when available (limited, particularly for generics); consult specific product labeling.

Solution, ophthalmic:

Paremyd: Hydroxyamphetamine hydrobromide 1% and tropicamide 0.25% (15 mL) [contains benzalkonium chloride]


Drug Interactions

There are no known significant interactions.


Monitoring Parameters

Ophthalmic exam, intraocular pressure, CNS reactions (especially in pediatric patients).


Adverse Reactions


Frequency not defined. Reported with Paremyd or similar medications.

Cardiovascular: Hypotension, myocardial infarction, tachycardia, vasomotor collapse, ventricular fibrillation

Central nervous system: Behavioral problems, headache, psychosis

Dermatologic: Pallor

Gastrointestinal: Nausea, vomiting, xerostomia

Hypersensitivity: Hypersensitivity reaction

Neuromuscular & skeletal: Muscle rigidity

Ophthalmic: Blurred vision, increased intraocular pressure, photophobia, stinging of eyes (transient)


Warnings/Precautions


Concerns related to adverse effects:

- CNS effects: May cause drowsiness and/or blurred vision, which may impair physical or mental abilities; patients must be cautioned about performing tasks that require mental alertness (eg, operating machinery, driving).

- Increased intraocular pressure: May cause a transient increase in intraocular pressure; use with caution in patients with glaucoma.

Disease-related concerns:

- Cardiovascular disease: Use caution in patients with hypertension, arrhythmias, or ischemic disease; monitor following administration.

- Diabetes: Use caution in patients with diabetes; monitor following administration.

- Thyroid disease: Use caution in patients with hyperthyroidism; monitor following administration.

Special populations:

- Contact lens wearers: May contain benzalkonium chloride, which may be adsorbed by contact lenses; remove contacts prior to administration and wait 15 minutes before reinserting.

- Elderly: Use with caution in the elderly; monitor closely for increased intraocular pressure following use.

- Pediatric: Use with caution in infants and children; may cause potentially dangerous CNS disturbances. Psychotic reactions, behavioral disturbances, and vasomotor or cardiorespiratory collapse in children have been reported with the use of anticholinergic drugs.

Other warnings/precautions:

- Appropriate use: For topical ophthalmic use only. To avoid excessive systemic absorption, apply gentle finger pressure to lacrimal sac for 2 to 3 minutes following application. Do not touch dropper tip to eyelids or any surface.


Pregnancy Risk Factor

C


Pregnancy Considerations

Animal reproduction studies have not been conducted with this combination. If ophthalmic agents are needed during pregnancy, the minimum effective dose should be used in combination with punctual occlusion to decrease potential exposure to the fetus (Samples, 1988).


Actions


Pharmacology

Hydroxyamphetamine hydrobromide is an indirect acting sympathomimetic agent which causes the release of norepinephrine from adrenergic nerve terminals, resulting in mydriasis. Tropicamide is a parasympatholytic agent which produces mydriasis and paralysis by blocking the sphincter muscle in the iris and the ciliary muscle.


Onset of Action

15 minutes


Time to Peak

60 minutes


Duration of Action

3 hours; complete recovery usually occurs in 6-8 hours, but may take up to 24 hours


Patient and Family Education


Patient Education

- Discuss specific use of drug and side effects with patient as it relates to treatment. (HCAHPS: During this hospital stay, were you given any medicine that you had not taken before? Before giving you any new medicine, how often did hospital staff tell you what the medicine was for? How often did hospital staff describe possible side effects in a way you could understand?)

- Educate patient about signs of a significant reaction (eg, wheezing; chest tightness; fever; itching; bad cough; blue skin color; seizures; or swelling of face, lips, tongue, or throat). Note: This is not a comprehensive list of all side effects. Patient should consult prescriber for additional questions.

Intended Use and Disclaimer: Should not be printed and given to patients. This information is intended to serve as a concise initial reference for healthcare professionals to use when discussing medications with a patient. You must ultimately rely on your own discretion, experience and judgment in diagnosing, treating and advising patients.

Copyright © 2016 - 2017
Doctor123.org | Disclaimer